Synapedia

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Promethazine

Promethazine is a first-generation antihistamine with sedative properties. It primarily acts as an H1 receptor antagonist and additionally possesses anticholinergic and antidopaminergic effects. The substance is medically used for the treatment of nausea, allergies, and as a sedative. Due to its sedative effects and anticholinergic side effects, caution is advised.

Depressiva
Depressiva
H1-Rezeptor
Muskarinischer Acetylcholinrezeptor

Mechanism of Action

  • H1 antagonist
  • M1 antagonist

Names / Identifiers

IUPAC: Promethazine

promethazine
Proazamine
60-87-7
Diphergan
Protazine
Vallergine
Dimapp
Promethazin
Fargan
Procit

Mechanism of Action

Promethazin wirkt hauptsächlich als Antagonist am H1-Histaminrezeptor und hat auch anticholinerge Eigenschaften.

Effects

Sedierung
Antiemetisch
Antihistaminisch
Anticholinerg
Anxiolytisch

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteIndividual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak2-4 hours
NotesThe duration of action may vary depending on dose and individual response.
Onset20-60 minutes
Total6-12 hours
After EffectsVariable, may include drowsiness.

Risks & Warnings

Warnings

  • Glaucoma
  • Prostatic hyperplasia
  • Pregnancy

Known Risks

  • medium
  • Mögliche Nebenwirkungen umfassen Schläfrigkeit, Schwindel und anticholinerge Effekte.

Safer Use

  • Start at a low dose.
  • Do not combine with alcohol or other sedatives.
  • Be aware of possible allergic reactions.

Harm reduction tips do not replace medical advice.

Known Interactions

  • Alcohol
  • Benzodiazepines
  • Opioids

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesIn vielen Ländern ist Promethazin nur auf Rezept erhältlich.

Not legal advice. Status may change.

Entdecken

Ähnliche Substanzen

Basierend auf Substanzklasse, Rezeptoren, Wirkmechanismen und Wirkprofil.

Gemeinsame Wirkungsmuster

Wirkungen, die Promethazine mit verwandten Substanzen teilt.

sedierung
auch beiKratom