Translated automatically – community improvements welcome.
Etizolam
Etizolam is a thienodiazepine-like sedative with anxiolytic, hypnotic, and muscle-relaxant properties. It primarily acts as an agonist at the GABA-A receptor, leading to enhanced inhibitory neurotransmission in the central nervous system. Due to its pharmacological effects, it is therapeutically used for the treatment of anxiety disorders and sleep disturbances. The risk of dependence and withdrawal symptoms is moderate and should be considered with prolonged use.
Mechanism of Action
- GABA-A agonist
Names / Identifiers
IUPAC: Etizolam
Mechanism of Action
Etizolam acts as an agonist at the GABA-A receptor, resulting in enhanced inhibition of neuronal activity. This leads to anxiolytic, sedative, and muscle-relaxant effects.
Dosage
Individual sensitivity varies. Not a dosage recommendation.
Duration
Risks & Warnings
Warnings
- Pregnancy
- Breastfeeding
- Severe respiratory diseases
Known Risks
- medium
- Mögliche Abhängigkeit und Toleranzentwicklung bei längerem Gebrauch.
Safer Use
- Start at low doses.
- Do not combine with alcohol or other sedatives.
Harm reduction tips do not replace medical advice.
Known Interactions
- Alcohol
- Opioids
- Other benzodiazepines
This list is not exhaustive. Interactions can have unpredictable effects.
Legal Status
Not legal advice. Status may change.
Receptor Targets
GABA-A
Der GABA-A-Rezeptor ist ein ligandengesteuerter Chloridkanal und der wichtigste inhibitorische Rezeptor im zentralen Nervensystem. Er besitzt multiple allosterische Bindungsstellen für verschiedene Substanzklassen.
Entdecken
Ähnliche Substanzen
Basierend auf Substanzklasse, Rezeptoren, Wirkmechanismen und Wirkprofil.