Synapedia

Translated automatically – community improvements welcome.

Pentobarbital

Pentobarbital is a barbiturate with sedative, hypnotic, and anticonvulsant effects. It acts by enhancing GABA-A receptor-mediated inhibition in the central nervous system. Due to its narrow therapeutic window and high toxicity, there is a significant risk of overdose and dependence. The substance was previously used as a sleeping aid and for anesthesia, but is less commonly used today due to safer alternatives.

Depressiva
Depressiva
GABA-A-Rezeptoren

Mechanism of Action

  • GABA-A receptor potentiation

Names / Identifiers

IUPAC: Pentobarbital

pentobarbital
Pentobarbitone
Nembutal
Mebubarbital
Pentobarbituric acid
Ethaminal
Dorsital
Mebumal
76-74-4
Rivadorm

Mechanism of Action

Pentobarbital verstärkt die GABA-A-Rezeptor-vermittelte Hemmung im zentralen Nervensystem, was zu sedierenden und hypnotischen Effekten führt.

Effects

sedierend
hypnotisch
antikonvulsiv
muskelrelaxierend
anxiolytisch

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteIndividual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak1-2 hours
NotesDuration of effect may vary depending on dose and individual metabolism.
Onset15-30 minutes
Total4-6 hours
After Effects2-4 hours

Risks & Warnings

Warnings

  • Respiratory diseases
  • Liver diseases
  • Pregnancy

Known Risks

  • high
  • Hohe Toxizität und Risiko für Überdosierung.

Safer Use

  • Start at a low dose
  • Avoid polydrug use with other depressants
  • Regular monitoring during use

Harm reduction tips do not replace medical advice.

Known Interactions

  • Alcohol
  • Benzodiazepines
  • Opioids

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesIn vielen Ländern ist Pentobarbital aufgrund seines Missbrauchspotenzials streng reguliert.

Not legal advice. Status may change.