Synapedia

Translated automatically – community improvements welcome.

Lofexidine

Lofexidine is a selective alpha-2 adrenergic receptor agonist primarily used for alleviating withdrawal symptoms in opioid dependence. It acts by inhibiting norepinephrine release, thereby reducing sympathetic overactivity. The substance has sedative and antihypertensive properties and is medically used to assist in withdrawal.

Alpha-2-Adrenozeptor-Agonisten

Mechanism of Action

  • Alpha-2 adrenergic agonist

Names / Identifiers

IUPAC: Lofexidine

Lofexidin
Lofexidine
Lofexidin HCl

Effects

Sedierung
Blutdrucksenkung
Reduktion von Entzugssymptomen
Verminderung von Angst
Entspannung

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteIndividual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak2-4 hours
NotesThe duration of action may vary depending on individual metabolism.
Onset1-2 hours
Total6-12 hours
After EffectsVariable

Risks & Warnings

Warnings

  • Severe cardiovascular diseases
  • Hypotension
  • Allergy to lofexidine

Known Risks

  • medium
  • Mögliche Nebenwirkungen umfassen Hypotonie, Sedierung und Bradykardie.

Safer Use

  • Start at a low dose.
  • Regular monitoring of blood pressure.
  • Avoid alcohol and other sedating substances.

Harm reduction tips do not replace medical advice.

Known Interactions

  • Antihypertensives
  • Sedatives
  • Opioids

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesLofexidin ist in vielen Ländern zur Behandlung von Opioidentzug zugelassen.

Not legal advice. Status may change.

Entdecken

Ähnliche Substanzen

Basierend auf Substanzklasse, Rezeptoren, Wirkmechanismen und Wirkprofil.

Gemeinsame Wirkungsmuster

Wirkungen, die Lofexidine mit verwandten Substanzen teilt.

entspannung
auch beiKratom, MDMA
sedierung
auch beiKratom