Translated automatically – community improvements welcome.
Butorphanol
Butorphanol is a synthetic opioid with partial agonist activity at μ-opioid receptors and agonist activity at κ-opioid receptors. It is primarily used for the treatment of moderate to severe pain. Due to its mechanism of action, it can cause side effects such as sedation and nausea. The potential for dependence is considered moderate, which is why cautious use is recommended.
Mechanism of Action
- κ-opioid agonist
- μ-opioid partial agonist
Names / Identifiers
IUPAC: Butorphanol
Mechanism of Action
Butorphanol wirkt als partieller Agonist am μ-Opioid-Rezeptor und als Agonist am κ-Opioid-Rezeptor, was zu schmerzlindernden Effekten führt.
Effects
Effects described from scientific sources. Individual experiences vary.
Dosage
Individual sensitivity varies. Not a dosage recommendation.
Duration
Risks & Warnings
Warnings
- Pregnancy
- Respiratory diseases
- severe liver or kidney diseases
Known Risks
- medium
- Mögliche Nebenwirkungen umfassen Sedierung und Übelkeit. Risiko einer Abhängigkeit.
Safer Use
- Start at low doses
- Avoid polydrug use with other sedatives
- Take regular breaks
Harm reduction tips do not replace medical advice.
Known Interactions
- Benzodiazepines
- Alcohol
- other opioids
This list is not exhaustive. Interactions can have unpredictable effects.
Legal Status
Not legal advice. Status may change.
Entdecken
Ähnliche Substanzen
Basierend auf Substanzklasse, Rezeptoren, Wirkmechanismen und Wirkprofil.