Synapedia

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N,N-dimethyl-3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-hep…

Cyclobenzaprine is a centrally acting muscle relaxant that is structurally related to tricyclic antidepressants. It primarily acts by inhibiting alpha2-adrenergic receptors and possesses anticholinergic properties. The substance is used to treat muscle spasms and can induce sedative effects. Side effects may include dry mouth, drowsiness, and cardiovascular effects.

Muskelrelaxantien

Mechanism of Action

  • alpha2-adrenergic inhibition
  • anticholinergic activity

Names / Identifiers

IUPAC: Cyclobenzaprine

Mechanism of Action

Cyclobenzaprin wirkt als Muskelrelaxans, indem es die zentrale Hemmung von spinalen Reflexen fördert und die serotonergen und noradrenergen Systeme beeinflusst.

Effects

Muskelrelaxation
Sedierung
Schmerzlinderung
Verminderung von Muskelspasmen
Anticholinerge Effekte

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteConsider individual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak3-6 hours
NotesEffect may vary depending on individual sensitivity.
Onset1-2 hours
Total12-24 hours
After EffectsFatigue, dizziness

Risks & Warnings

Warnings

  • Acute myocardial infarction
  • Hyperthyroidism
  • Glaucoma

Known Risks

  • medium
  • Kann Schläfrigkeit, Schwindel und anticholinerge Effekte verursachen.

Safer Use

  • Avoid alcohol and other sedating substances.
  • Do not drive if you feel drowsy.

Harm reduction tips do not replace medical advice.

Known Interactions

  • MAO inhibitors
  • other CNS depressants

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesIn vielen Ländern ist Cyclobenzaprin nur auf Rezept erhältlich.

Not legal advice. Status may change.

Entdecken

Ähnliche Substanzen

Basierend auf Substanzklasse, Rezeptoren, Wirkmechanismen und Wirkprofil.

Gemeinsame Wirkungsmuster

Wirkungen, die N,N-dimethyl-3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-hep… mit verwandten Substanzen teilt.

schmerzlinderung
auch beiSSRI, Kratom, Ketamin
sedierung
auch beiKratom