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Azaperone

Azaperon is a typical neuroleptic from the group of butyrophenones, primarily used as a sedative and antipsychotic. It mainly acts by blocking dopamine D2 receptors and additionally has antagonistic effects on alpha-1 adrenergic receptors. In veterinary medicine, it is frequently used to calm animals. The substance can induce sedative effects and carries risks such as extrapyramidal symptoms and cardiovascular side effects.

Neuroleptika

Mechanism of Action

  • Alpha-1-Adrenozeptor-Antagonist
  • Dopamin-D2-Rezeptor-Antagonist

Names / Identifiers

IUPAC: Azaperone

Mechanism of Action

Azaperone wirkt als Antagonist an Dopamin- und Serotoninrezeptoren, was zu einer sedierenden und anxiolytischen Wirkung führt.

Effects

sedierend
anxiolytisch
antipsychotisch
muskelrelaxierend
antidepressiv

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteIndividual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak2-4 hours
NotesThe duration of action may vary depending on dose and individual metabolism.
Onset30-60 minutes
Total6-12 hours
After EffectsVariable

Risks & Warnings

Warnings

  • Do not use in case of known hypersensitivity to butyrophenones.
  • Caution in patients with cardiovascular diseases.

Known Risks

  • medium
  • Mögliche Nebenwirkungen umfassen Sedierung, extrapyramidale Symptome und kardiovaskuläre Effekte.

Safer Use

  • Start at a low dose.
  • Consider regular medical check-ups.

Harm reduction tips do not replace medical advice.

Known Interactions

  • May interact with other central depressants.

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesIn der Veterinärmedizin häufig verwendet.

Not legal advice. Status may change.