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Amitriptyline

Amitriptyline is a tricyclic antidepressant that primarily works by inhibiting the reuptake of serotonin and norepinephrine. It also possesses antagonistic effects at various receptors, leading to sedative and anticholinergic effects. The substance is used not only for the treatment of depression but also for pain therapy. Due to its side effect profile and toxic potential in overdose, a moderate risk profile should be considered.

Antidepressiva

Mechanism of Action

  • NET inhibitor
  • SERT inhibitor

Names / Identifiers

IUPAC: Amitriptyline

Mechanism of Action

Amitriptylin wirkt hauptsächlich durch die Hemmung der Wiederaufnahme von Serotonin und Noradrenalin in die präsynaptischen Neuronen, was zu einer erhöhten Verfügbarkeit dieser Neurotransmitter im synaptischen Spalt führt.

Effects

Antidepressiv
Schmerzlindern
Sedierend
Angstlösend
Anticholinerg
Appetitanregend
Müdigkeit
Kognitive Beeinträchtigung

Effects described from scientific sources. Individual experiences vary.

Dosage

Safety NoteConsider individual variation, start at a low dose, no medical advice.

Individual sensitivity varies. Not a dosage recommendation.

Duration

Peak4-6 hours
NotesEffect may vary depending on individual metabolism.
Onset1-3 hours
Total24 hours
After Effects12-24 hours

Risks & Warnings

Warnings

  • Pregnancy
  • Heart diseases
  • Glaucoma

Known Risks

  • medium
  • Mögliche Nebenwirkungen umfassen Sedierung, anticholinerge Effekte und kardiovaskuläre Risiken.

Safer Use

  • Start at a low dose
  • Regular medical check-ups
  • Avoid alcohol and other sedatives

Harm reduction tips do not replace medical advice.

Known Interactions

  • MAO inhibitors
  • Alcohol
  • Benzodiazepines

This list is not exhaustive. Interactions can have unpredictable effects.

Legal Status

ATVerschreibungspflichtig
CHVerschreibungspflichtig
DEVerschreibungspflichtig
USVerschreibungspflichtig
NotesAmitriptylin ist in vielen Ländern als verschreibungspflichtiges Medikament eingestuft.

Not legal advice. Status may change.